Brønsted-Acid Catalyzed Diastereo- and Enantioselective Synthesis of Spiroisoindolinones from Enamides.

 0 Người đánh giá. Xếp hạng trung bình 0

Tác giả: Leon Donner, Miro Halaczkiewicz, Harald Kelm, Georg Manolikakes, Arianit Maraj, Mareike Riedel

Ngôn ngữ: eng

Ký hiệu phân loại: 296.127 Specific types of Talmudic literature

Thông tin xuất bản: Germany : Chemistry (Weinheim an der Bergstrasse, Germany) , 2025

Mô tả vật lý:

Bộ sưu tập: NCBI

ID: 176170

 A highly stereoselective Brønsted-acid catalyzed synthesis of densely substituted spiroisoindolinones from enamides and 3-hydroxy-isoindolinones is described. With simple Brønsted-acids, such as para-toluene sulfonic acid, spiroisoindolinones with three contiguous stereogenic centers are formed in high yields (up to 97 %) and diastereoselectivities (up to >
 98 : <
 2 : 0 : 0 dr) under mild reaction conditions. With the use of a chiral phosphoric acid catalyst, a diastereo- and enantioselective synthesis of the corresponding spiroisoindolinones was achieved. Mechanistic investigations indicate a step-wise mechanism via an initial addition of the enamide to an electrophilic N-acylimine species followed by an intramolecular aza-Friedel-Crafts reaction. Addition of a strong Lewis acid can be used to facilitate the second step for less reactive substrates.
Tạo bộ sưu tập với mã QR

THƯ VIỆN - TRƯỜNG ĐẠI HỌC CÔNG NGHỆ TP.HCM

ĐT: (028) 36225755 | Email: tt.thuvien@hutech.edu.vn

Copyright @2024 THƯ VIỆN HUTECH