Total Synthesis of DMOA-Derived Meroterpenoids: Achieving Selectivity in the Synthesis of (+)-Berkeleyacetal D and (+)-Peniciacetal I.

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Tác giả: Chao Li, Xiaotong Luo, Jianpeng Zhang, Jingfu Zhang

Ngôn ngữ: eng

Ký hiệu phân loại: 594.38 *Pulmonata

Thông tin xuất bản: United States : Journal of the American Chemical Society , 2025

Mô tả vật lý:

Bộ sưu tập: NCBI

ID: 191373

The synthesis of complex natural products requires efficient control over chemoselectivity, stereoselectivity, and regioselectivity. Berkeleyacetals, a subfamily of 3,5-dimethylorsellinic acid (DMOA)-derived meroterpenoids, pose substantial synthetic challenges due to their densely functionalized and highly oxidized architectures, which have constrained synthetic efforts. Here, we present the first total synthesis of this class of DMOA-derived meroterpenoids, specifically (+)-berkeleyacetal D and (+)-peniciacetal I. Our approach features a chemoselective deprotonation followed by an intramolecular single-electron transfer (SET) from an enolate to an alkyl bromide, enabling the construction of the 2,3-dihydrofuran ring in berkeleyacetal D. Additional selective transformations include an
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