A robust fluorogenic substrate for chikungunya virus protease (nsP2) activity.

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Tác giả: Cedric Bobst, Matthew Bogyo, Shruti Choudhary, Marcin Drag, Jasna Fejzo, Chenzhou Hao, Jeanne A Hardy, Michael Z Lin, Sparsh Makhaik, Wioletta Rut, Paul Thompson, Tulsi Upadhyay, Michael Westberg, Euna Yoo

Ngôn ngữ: eng

Ký hiệu phân loại: 343.09482 Military, defense, public property, public finance, tax, commerce (trade), industrial law

Thông tin xuất bản: United States : Protein science : a publication of the Protein Society , 2025

Mô tả vật lý:

Bộ sưu tập: NCBI

ID: 239960

Chikungunya virus (CHIKV) is an emerging pathogen with pandemic potential. CHIKV infection in humans is transmitted by mosquitoes and induces common symptoms of high fever, arthralgia and myalgia. Because no specific antiviral drugs for treatment of CHIKV infection are available, drug development remains a central goal. The chikungunya virus protease from nsP2 (CHIKVP) has emerged as a key drug target due to its indispensable role in viral replication via cleavage of the viral polyprotein. To date, effective tools for screening for CHIKVP inhibitors that reflect the most critical polyprotein cleavage sites have been lacking, hampering drug-development efforts. We found that the recognition ability of CHIKVP is sensitive to the length of peptide substrates. In this study, we report a robust fluorogenic substrate comprising a 15-mer peptide derived from the nsP3/4 junction from the CHIKV polyprotein. This peptide is flanked by an ACC-Lys(dnp) donor-quencher pair. Our new substrate acc-CHIK
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