Identification and optimization of a small molecule inhibitor of the ovarian tumor protease of the Crimean-Congo hemorrhagic fever virus.

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Tác giả: Lorenz Beckmann, Maik Icker, Fabian Liessmann, Jens Meiler, Dominic Rieger, Michael Schaefer, Phillip Schlegel, Clara T Schoeder, Maik Tretbar, Nicole Urban

Ngôn ngữ: eng

Ký hiệu phân loại:

Thông tin xuất bản: England : Bioorganic & medicinal chemistry , 2025

Mô tả vật lý:

Bộ sưu tập: NCBI

ID: 497744

Crimean-Congo hemorrhagic fever (CCHF) is a viral tick-borne disease with fatality rates of up to 30 %. Currently, there are no vaccines or specific antivirals available. The genome of the CCHF virus (CCHFV) encodes an ovarian tumor (OTU) protease with a deubiquitinating activity that is responsible for the evasion of the innate immune response. Therefore, the inhibition of the OTU protease could provide a strategy for the treatment of CCHFV infections. In this study, we screened for small-molecule inhibitors of CCHFV OTU using a fluorescent ubiquitin rhodamine 110 assay. We identified and validated a 2-aminothiazole hit compound (IC
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