Fabrication of lipid-modified drug nanocrystals loaded injectable hydrogel for breast cancer therapy.

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Tác giả: Kanchan Bharti, Pooja Goswami, Abhishek Jha, Biplob Koch, Manish Kumar, Manjit Manjit, Brahmeshwar Mishra, Ritika Srivastava

Ngôn ngữ: eng

Ký hiệu phân loại: 005.742 *Data dictionaries and directories

Thông tin xuất bản: Switzerland : Discover nano , 2025

Mô tả vật lý:

Bộ sưu tập: NCBI

ID: 66005

The current study includes the design of soluplus stabilized, lipid-coated, and fucoidan-oleylamine conjugate modified paclitaxel nanocrystals. The nanocrystals (Lipid-NCs) were about 100 nm, homogeneous, stable and showed improved drug release compared to pure PTX. The nanocrystals were subsequently loaded in an in situ gel-forming hydrogel for the intratumoral injection. The resulting hydrogel exhibited a sol-form at the lower temperature of 2-8 °C while converted to a gel-form at the body temperature. The injectable hydrogel had a reasonable viscosity, an acceptable pH, good syringeability, and a quick sol-gel transition. The hydrogel demonstrated high payload potential, homogeneous distribution, and controlled long-term drug release. In vivo studies revealed the higher efficacy of Lipid-NCs hydrogel in tumor inhibition while avoiding systemic toxicity, compared to pure PTX-loaded hydrogel and intravenously administered PTX. In conclusion, nanocrystal-loaded hydrogel is a promising localized drug delivery system for breast cancer therapy.
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