Antitumor efficacy of intermittent low-dose erlotinib plus sulindac via MHC upregulation and remodeling of the immune cell niche.

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Tác giả: Powel H Brown, Roderick H Dashwood, Wan Mohaiza Dashwood, Melek Demirhan, Yunus Demirhan, Sabeeta Kapoor, Altaf Mohammed, Ahmed Muhsin, Praveen Rajendran, Michelle I Savage, Shizuko Sei, Alessandro Shapiro, Krishna M Sinha, Jacklyn Thompson, Jorge E Tovar Perez, Chakrapani Tripathi, Eduardo Vilar, Mahira Zaheer

Ngôn ngữ: eng

Ký hiệu phân loại:

Thông tin xuất bản: United States : International journal of cancer , 2025

Mô tả vật lý:

Bộ sưu tập: NCBI

ID: 699244

 A previously reported clinical trial in familial adenomatous polyposis (FAP) patients treated with erlotinib plus sulindac (ERL + SUL) highlighted immune response/interferon-γ signaling as a key pathway. In this study, we combine intermittent low-dose ERL ± SUL treatment in the polyposis in rat colon (Pirc) model with mechanistic studies on tumor-associated immune modulation. At clinically relevant doses, short-term (16 weeks) and long-term (46 weeks) ERL ± SUL administration results in near-complete tumor suppression in Pirc colon and duodenum (p <
  0.0001). We identify a low-dose threshold for significant antitumor activity in Pirc rats given SUL at 125 ppm in the diet plus ERL at 5 mg/kg body weight via twice-weekly oral gavage (SUL125 + ERL5 × 2). Longitudinal analyses show diminished expression of MHC class I and II genes in polyps larger than Grade 5, a novel finding in the Pirc model. Treatment with ERL ± SUL upregulates the corresponding MHC and immune-associated factors in a subset of Pirc colon polyps, Pirc tumor cell lines, murine colon carcinoma cells, and FAP patient-derived organoids, with Nlrc5 playing a critical role in this effect. Imaging mass cytometry reveals that SUL125 + ERL5 × 2 increases tumor-associated Cd4
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