Design and synthesis of novel cyclohexanecarboxamides with anticonvulsant effect by activating Nrf2-ARE pathway.

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Tác giả: Walaa H Abd-Allah, Mohammed S Abdel-Maksoud, Marawan A Elbaset, Rasha M Hassan, Ibrahim M Ibrahim, Reda M S Korany

Ngôn ngữ: eng

Ký hiệu phân loại: 944.08 1870

Thông tin xuất bản: United States : Bioorganic chemistry , 2025

Mô tả vật lý:

Bộ sưu tập: NCBI

ID: 713602

This study investigated a series of novel cyclohexanecarboxamide derivatives 4a-e, 5a-e and 6a-e as anticonvulsant and neuroprotective agents. Compounds 4a-e, 5a-e, and 6a-e were synthesized starting from cyclohexanone and aniline derivatives and evaluated for their anticonvulsant effects using maximal electroshock (MES) and subcutaneous pentylenetetrazole (scPTZ) seizure models. The most potent compounds 4b, 5c, and 6d demonstrated 83.33 % protection in the scPTZ test, while compounds 5a and 6b showed 100 % protection in the MES test. Further quantitative evaluation showed that compound 6d was the most active derivative in scPTZ test (ED
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