Pyruvate metabolism enzyme DLAT promotes tumorigenesis by suppressing leucine catabolism.

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Tác giả: Ziyi Cao, Suzhen Chen, Xuefeng Dou, Yunqing Gu, Liu Han, Quanxin Jiang, Fuming Li, Hongtao Li, Huimin Li, Junli Liu, Sijia Lu, Hai-Long Piao, Qiqi Qian, Haipeng Sun, Mijia Tao, Ning Wang, Wei Wang, Junting Xu, Yingjie Xu, Weiwei Yang, Hanrui Yin, Limin Yin, Xianjing Zhang, Liaoyuan Zheng, Peihui Zhou, Qian Zhou

Ngôn ngữ: eng

Ký hiệu phân loại: 746.445 *Applique

Thông tin xuất bản: United States : Cell metabolism , 2025

Mô tả vật lý:

Bộ sưu tập: NCBI

ID: 726893

Pyruvate and branched-chain amino acid (BCAA) metabolism are pivotal pathways in tumor progression, yet the intricate interplay between them and its implications for tumor progression remain elusive. Our research reveals that dihydrolipoamide S-acetyltransferase (DLAT), a pyruvate metabolism enzyme, promotes leucine accumulation and sustains mammalian target of rapamycin (mTOR) complex activation in hepatocellular carcinoma (HCC). Mechanistically, DLAT directly acetylates the K109 residue of AU RNA-binding methylglutaconyl-coenzyme A (CoA) hydratase (AUH), a critical enzyme in leucine catabolism, inhibiting its activity and leading to leucine accumulation. Notably, DLAT upregulation correlates with poor prognosis in patients with HCC. Therefore, we developed an AUH
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