The importance role of central proline to the antimicrobial potency and selectivity of indolicidin.

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Tác giả: Le Minh Bui, Thinh Pham Duc, Hai Bui Thi Phuong, Tung Truong Thanh, Hang Ngo Thu, Linh Dang Thuy, Hoa Ngo Van, Khanh Hoang Van, Mao Can Van, Tan Nguyen Van, Khoa Nguyen Vu, Huy Luong Xuan

Ngôn ngữ: eng

Ký hiệu phân loại:

Thông tin xuất bản: Germany : Archives of microbiology , 2025

Mô tả vật lý:

Bộ sưu tập: NCBI

ID: 727717

The increasing prevalence of multidrug-resistant pathogens urged the development of new therapeutic strategies, and antimicrobial peptides (AMPs) have emerged as promising candidates. Indolicidin, a proline-rich AMP, is effective against a wide range of pathogens by penetrating the membrane to disrupt the cytoplasmic membrane or inhibit DNA synthesis. This study investigates the impact of replacing the central proline residue in Indolicidin with glycine (IND-7G), D-proline (IND-7DP), or lysine (IND-7K). Results show that both glycine and D-proline substitutions significantly reduced antimicrobial activity with lower hemolysis than the parent peptide. Besides, the analog having lysine substitution (IND-7K) slightly increased activity against E. coli and C. albicans but reduced potency against S. aureus, E. faecalis, and K. pneumoniae. The hemolytic activity of IND-7K remained comparable to that of Indolicidin. These findings demonstrated the essential role of proline in maintaining the antimicrobial efficacy of Indolicidin.
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