Targeting the Dependence on PIK3C3-mTORC1 Signaling in Dormancy-Prone Breast Cancer Cells Blunts Metastasis Initiation.

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Tác giả: Julio A Aguirre-Ghiso, James V Alvarez, Stéphane Angers, Virginie Calderon, Jean-François Côté, Stanislav Drapela, Islam E Elkholi, Ana P Gomes, Steven Hébert, Claudia L Kleinman, Hellen Kuasne, Graham Macleod, Camille Malouf, Alain Pacis, Morag Park, Amélie Robert, Joshua L Wu

Ngôn ngữ: eng

Ký hiệu phân loại: 597.9257 Reptilia (Reptiles)

Thông tin xuất bản: United States : Cancer research , 2025

Mô tả vật lý:

Bộ sưu tập: NCBI

ID: 746002

Halting breast cancer metastatic relapse following primary tumor removal remains challenging due to a lack of specific vulnerabilities to target during the clinical dormancy phase. To identify such vulnerabilities, we conducted genome-wide CRISPR screens on two breast cancer cell lines with distinct dormancy properties: 4T1 (short-term dormancy) and 4T07 (prolonged dormancy). The dormancy-prone 4T07 cells displayed a unique dependency on class III PI3K (PIK3C3). Unexpectedly, 4T07 cells exhibited higher mechanistic target of rapamycin complex 1 (mTORC1) activity than 4T1 cells due to lysosome-dependent signaling occurring at the cell periphery. Pharmacologic inhibition of PIK3C3 suppressed this phenotype in the 4T1-4T07 models as well as in human breast cancer cell lines and a breast cancer patient-derived xenograft. Furthermore, inhibiting PIK3C3 selectively reduced metastasis burden in the 4T07 model and eliminated dormant cells in a HER2-dependent murine breast cancer dormancy model. These findings suggest that PIK3C3-peripheral lysosomal signaling to mTORC1 may represent a targetable axis for preventing dormant cancer cell-initiated metastasis in patients with breast cancer. Significance: Dormancy-prone breast cancer cells depend on the class III PI3K to mediate peripheral lysosomal positioning and mTORC1 hyperactivity, which can be targeted to blunt breast cancer metastasis.
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