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Spirocyclic compounds as innovative tools in drug discovery for medicinal chemists
Tác giả: Marina T Varela, Gleiston G Dias, Luiz Fernando N de Oliveira, Ramon G de Oliveira, Francielle D Aguiar, João Pedro Nogueira, Luiza R Cruz, Luiz C Dias
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc: 
 
Spirocyclic compounds as innovative tools in drug discovery for medicinal chemists
Tác giả: Marina T Varela, Gleiston G Dias, Luiz Fernando N de Oliveira, Ramon G de Oliveira, Francielle D Aguiar, João Pedro Nogueira, Luiza R Cruz, Luiz C Dias
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc: 
 
Design, synthesis, and biological evaluation of quinazolinone-dihydropyrimidinone as a potential anti-diabetic agent via...
Tác giả: Arvind Kumar Jaiswal, Ajay Kishor Kushawaha, Akhilesh K Tamrakar, Koneni V Sashidhara, Pawan Kumar, Alisha Ansari, Nikita Chhikara, Hemlata Bhatt, Sarita Katiyar, Ishbal Ahmad, Abhijit Deb Choudhury, Rabi Sankar Bhatta
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc: 
 
Design, synthesis, and biological evaluation of novel quinoline carboxylic acid based styryl/alkyne hybrid molecule as a...
Tác giả: Richa Singh, Vinita Kushwaha, Vishal M Balaramnavar, Rabi Sankar Bhatta, Ravindra Kumar, Anil N Gaikwad, Arun K Sinha, Sumit K Rastogi, Prashant Rai, Santosh Kumar, Nilesh Khandelwal, Sanchita Gupta, Amol Chhatrapati Bisen, Salil Varshney, Astha Singh
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc: 
 
Corrigendum to "A chemical modification of a peroxisome proliferator-activated receptor pan agonist produced a shift to ...
Tác giả: Antonio Laghezza, Carmen Cerchia, Leonardo Brunetti, Luca Piemontese, Paolo Tortorella, Abanish Biswas, Ravi Pratap Singh, Suhas Tambe, C A Sudeep, Ashok Kumar Pattnaik, Venkatesan Jayaprakash, Paolo Paoli, Massimo Genovese, Antonio Lavecchia, Fulvio Loiodice, Roberta Montanari, Davide Capelli, Judith Wackerlig, Stefan Simic, Emanuele Falbo, Lucia Pecora, Rosalba Leuci
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc: 
 
Design, synthesis, and biological evaluation of β-carboline derivatives as ABCB1 inhibitors for reversing multidrug resi...
Tác giả: Yuanyuan Wang, Nanjin Ding, Yunpeng Zhao, Fengqing Wang, Wen Liu, Zhe Chen, Weiguang Sun, Lianghu Gu, Yonghui Zhang
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc: 
 
Discovery of β-amino acid substituted naphthalene sulfonamide derivatives as potent Kelch-like ECH-associated protein 1-...
Tác giả: Ziquan Zhao, Hongjin Lu, Junjie Wang, Tingting Wu, Shicheng Xu, Yuxin Ge, Qidong You, Zhengyu Jiang, Mengchen Lu
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc: 
 
Discovery of highly potent dual GSPT1/BRD4 degraders with anti-AML activity
Tác giả: Yue Xu, Hang Yang, Jie Fu, Qinrong Lin, Chunhong Chen, Ningning Shi, Jianping Cai, Ke Li, Shuanghu Wang, Ruijuan Gao, Dapeng Dai, Yunxuan Li, Yuying Qi, Fangling Zhao, Yun Hong, Binbin Cheng, Zebei Lu, Jiaming Zhang, Chunyi Guo
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc: 
 
Discovery of a novel Wnt inhibitor DK419: Reversing temozolomide resistance in glioblastoma by switching off Wnt/β-caten...
Tác giả: Peiying Bai, Peng Wang, Ting Ren, Qing Tang, Na Zhang, Lijiao Zhao, Rugang Zhong, Guohui Sun
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc: 
 
Natural pyrrolo[1,2-a]quinazolinone derivatives: Design, synthesis, characterization, and bio-evaluation as novel antivi...
Tác giả: Yanhong Wei, Fuqiang Zheng, Mengmeng Kong, Shaoyong Ke, Lirong Guo, Wenxuan Chen, Hexiang Wang, Longzhu Bao, Zhaoyuan Wu, Ying Li, W Alateng, Jianglong Su
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc: 
 
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