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31-40 trong số 230 kết quả
Corrigendum to "A chemical modification of a peroxisome proliferator-activated receptor pan agonist produced a shift to ...
Tác giả: Antonio Laghezza, Carmen Cerchia, Leonardo Brunetti, Luca Piemontese, Paolo Tortorella, Abanish Biswas, Ravi Pratap Singh, Suhas Tambe, C A Sudeep, Ashok Kumar Pattnaik, Venkatesan Jayaprakash, Paolo Paoli, Massimo Genovese, Antonio Lavecchia, Fulvio Loiodice, Roberta Montanari, Davide Capelli, Judith Wackerlig, Stefan Simic, Emanuele Falbo, Lucia Pecora, Rosalba Leuci
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  709.012
 
Ascertaining a Structural Basis in Drug Discovery and Development
Tác giả: David E Heppner
Xuất bản: United States: Journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  571.876
 
Discovery of Potent and Brain-Penetrant Bicyclic NLRP3 Inhibitors with Peripheral and Central In Vivo Activity
Tác giả: Oscar Mammoliti, Rodrigo Carbajo, Santiago Cañellas, Saskia De Hoog, Samuël Demin, Harrie J M Gijsen, Geerwin Hache, Tom Jacobs, Soufyan Jerhaoui, Joseph Leenaerts, Ferdinand H Lutter, Michel Mahieu, Laura Perez-Benito, Rosalie Matico, Robyn Miller, Daniel Oehlrich, Mathieu Perrier, Pavel Ryabchuk, Wim Schepens, Sujata Sharma, Marijke Somers, Javier Suarez, Michel Surkyn, Xiaodi Yu, Nina Van Opdenbosch, Tinne Verhulst, Astrid Bottelbergs, Marion L C Prieri, Leonardo Bontempi, Sofie Embrechts, Ine Paesmans, Michela Bassi, Anindya Bhattacharya
Xuất bản: United States: Journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  612.826
 
Discovery of Novel Aromatic Urea-Imidazole Salt Derivatives for Cancer Therapy via Targeting ERK1/2
Tác giả: Mengqi Wang, Shuping Yang, Xinge Li, Yingying Zheng, Yan Bai, Wenhan Luo, Gongming Zhu, Junbiao Chang, Bo Zhu
Xuất bản: United States: Journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  332.6457
 
Discovery of Novel Isoxazole-Based Small-Molecule Toll-Like Receptor 8 Antagonists
Tác giả: Troy Matziol, Valerij Talagayev, Tjaša Slokan, Nika Strašek Benedik, Janine Holze, Matej Sova, Gerhard Wolber, Günther Weindl
Xuất bản: United States: Journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  372.427
 
Identification of Structurally Novel KRAS
Tác giả: David Huang, Francesco Manoni, Heejun Lee, Cui Li, Xun Li, Patricia Lopez, Vu Ma, Jose M Medina, Christopher Mohr, Olga A Mukhina, Alexander J Pickrell, John Stellwagen, Zhen Sun, Wenting Wu, Wenhan Zhang, Kai Zhu, Upendra P Dahal, Liaoyuan A Hu, Monica Leavitt, Wencui Li, Yu Li, Yingli Ma, Karen Rex, Rongfeng Liu, Anne Y Saiki, Paul Wang, Yaping Sun, Dongcheng Dai, Nuria A Tamayo, Brian A Lanman, Jennifer R Allen, Abhisek Banerjee, Victor J Cee, Josephine Eshon, Michael J Frohn, Matthew R Kaller
Xuất bản: United States: Journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  003.1
 
Design, synthesis, and biological evaluation of β-carboline derivatives as ABCB1 inhibitors for reversing multidrug resi...
Tác giả: Yuanyuan Wang, Nanjin Ding, Yunpeng Zhao, Fengqing Wang, Wen Liu, Zhe Chen, Weiguang Sun, Lianghu Gu, Yonghui Zhang
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  332.6457
 
Discovery of β-amino acid substituted naphthalene sulfonamide derivatives as potent Kelch-like ECH-associated protein 1-...
Tác giả: Ziquan Zhao, Hongjin Lu, Junjie Wang, Tingting Wu, Shicheng Xu, Yuxin Ge, Qidong You, Zhengyu Jiang, Mengchen Lu
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  668.43
 
Discovery of highly potent dual GSPT1/BRD4 degraders with anti-AML activity
Tác giả: Yue Xu, Hang Yang, Jie Fu, Qinrong Lin, Chunhong Chen, Ningning Shi, Jianping Cai, Ke Li, Shuanghu Wang, Ruijuan Gao, Dapeng Dai, Yunxuan Li, Yuying Qi, Fangling Zhao, Yun Hong, Binbin Cheng, Zebei Lu, Jiaming Zhang, Chunyi Guo
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  342.0854
 
Structure-Based Discovery of a Highly Selective, Oral Polo-Like Kinase 1 Inhibitor with Potent Antileukemic Activity
Tác giả: Jianyu Nie, Xiaojiao Sun, Yan He, Mingxin Zhu, Xinglong Zhang, Qin Wang, Zhenming Liu, Zhouling Xie, Zhongtang Li, Chenzhong Liao
Xuất bản: United States: Journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  796.353
 

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