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51-60 trong số 230 kết quả
One-Pot Synthesis of Novel Tetrasubstituted α-Aminophosphonates Derived from α-Methylphosphoserine and
Tác giả: Misael López-Castillo, Mario Ordóñez, Itzel Bernal-Evangelista, Gil A Vázquez-Arredondo, Martha Vanessa Gutiérrez-Baños, Ivan Romero-Estudillo, Gabriela Castañeda-Corral
Xuất bản: United States: Journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  615.322
 
Correction to "Development of BromoTag: A "Bump-and-Hole"-PROTAC System To Induce Potent, Rapid, and Selective Degradati...
Tác giả: Adam G Bond, Conner Craigon, Kwok-Ho Chan, Andrea Testa, Athanasios Karapetsas, Rotimi Fasimoye, Thomas Macartney, J Julian Blow, Dario R Alessi, Alessio Ciulli
Xuất bản: United States: Journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  272.3
 
Discovery of novel imidazo[1,2-b]pyridazine derivatives as potent covalent inhibitors of CDK12/13
Tác giả: Meng Xia, Ziteng Li, Hong Ding, Mingliang Wang, Hanrui Jiang, Yuanqing Li, Linghao Hu, Yongchang He, Siqi Huang, Lei Tang, Cheng Luo, Shuangxi Gu
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  332.6457
 
Novel HOCl-Responsive Theranostic Prodrug for the Early Diagnosis and Therapy of Ischemic Stroke
Tác giả: Huayu Wang, Kemin Li, Linjie Zhang, Taihe Han, Shuai Mu, Youwei Song, Zehua Han, Haiyu Zhao, Xiaoyan Liu, Haixia Zhang
Xuất bản: United States: Journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  616.0757
 
Discovery of novel sitolactone derivative leading to PANoptosis and differentiation of acute myeloid leukemia cells
Tác giả: Jiefu Wang, Ning Wang, Guang Yang, Junfeng Wang, Shuangwei Liu, Kun Zhang, Mengmeng Wang, Ning Liu, Chenyang Wang, Ning Li, Linrong Mu, Yurui Jiang, Jia Chen, Jinxiao Li
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  616.99419
 
Development of potent indole-3-carboxamide autotaxin inhibitors with preferred lipophilicity for in vivo treatment of pu...
Tác giả: Deyi Ma, Nan Jiang, Jiachen Zhang, Hongrui Lei, Xin Zhai
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  612.647
 
Substitutions at the C-8 position of quinazolin-4-ones improve the potency of nicotinamide site binding tankyrase inhibi...
Tác giả: Chiara Bosetti, Dionysis Kampasis, Shoshy A Brinch, Albert Galera-Prat, Maria Karelou, Saurabh S Dhakar, Juho Alaviuhkola, Jo Waaler, Lari Lehtiö, Ioannis K Kostakis
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  949.5074
 
Discovery of Cationic Lugdunin Derivatives with Membrane-Disrupting Activity against Resistant Bacteria via Radical Reac...
Tác giả: Yuhang He, Jie Su, Hailong Zhang, Kairong Wang, Min Li, Muhammad S Fareed, Yixuan Ren, Panpan Wang, Zhaopeng Wang, Daicao Wan, Ting Ma, Wenjin Yan
Xuất bản: United States: Journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  641.62
 
Rational Design and Optimization of a Potent IDO1 Proteolysis Targeting Chimera (PROTAC)
Tác giả: Paige J Monsen, Prashant V Bommi, Michael Egozi, Sonam Jha, Sara F Dunne, Hong Jiang, Guiqin Song, Fang Zhang, Steven Kregel, Ali Vaziri-Gohar, Sean W Fanning, Pilar Sanchez-Gomez, Arabela A Grigorescu, Jacob M Allen, Bakhtiar Yamini, Rimas V Lukas, Derek A Wainwright, Gary E Schiltz, Kristen L Lauing, Yingyu Mao, Payton Berardi, Lijie Zhai, Oluwatomilayo Ojo, Manon Penco-Campillo, Taylor Koch
Xuất bản: United States: Journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  519.57
 
Rational design of dual-agonist peptides targeting GLP-1 and NPY2 receptors for regulating glucose homeostasis and body ...
Tác giả: Jing Liu, Weiwen Lu, Changhong Wei, Neng Jiang, Han Wu, Zhiming Yan, Yun Liu, Chunli Tang, Yangxin Chen, Shuang Wang, Weizhong Tang, Jing Han
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  211.7
 

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