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181-190 trong số 235 kết quả
Development of 3-arylaminothiophenic-2-carboxylic acid derivatives as new FTO inhibitors showing potent antileukemia act...
Tác giả: Deyan Zhang, Ze Dong, Xinyi Hu, Yue Huang, Ming Li, Lu Liu, Xiaomin Song, Zhen Wang, Wenyang Xia, Cai-Guang Yang, Xi Zhang
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  338.9
 
Novel thiazolones for the simultaneous modulation of PPARγ, COX-2 and 15-LOX to address metabolic disease-associated por...
Tác giả: Mai S El-Shoukrofy, Sherien A Abdelhady, Mahmoud A Agami, Ahmed S F Belal, Ali H Eid, Reem H Elhamammy, Ahmed F El-Yazbi, Perihan A Elzahhar, Azza Ismail, Monica S Makkar, Daniel Merk, Rasha Nassra, Hisham A Nematalla, Minh Sai, Ahmed Wahid
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  668.374
 
Discovery of novel tranylcypromine-indazole-based derivatives as LSD1 inhibitors for acute myeloid leukemia treatment
Tác giả: Ming-Jie Huang, Beiling Gao, Lihua Huang, Qiuge Liu, Jian Song, Saiyang Zhang
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  769.565
 
Design, synthesis and biological evaluation of diarylmethyl amine derivatives with anti-ulcerative colitis activity via ...
Tác giả: Zhongyang Ren, Xin Li, Guoyun Liu, Xiaotong Wang, Jie Yang, Xu Zhang
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  668.374
 
Design, synthesis, and biological evaluation of quinazolinone-dihydropyrimidinone as a potential anti-diabetic agent via...
Tác giả: Arvind Kumar Jaiswal, Ishbal Ahmad, Alisha Ansari, Rabi Sankar Bhatta, Nikita Chhikara, Abhijit Deb Choudhury, Hemlata Bhatt, Sarita Katiyar, Ajay Kishor Kushawaha, Pawan Kumar, Koneni V Sashidhara, Akhilesh K Tamrakar
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  378.242
 
Design, synthesis, and biological evaluation of novel quinoline carboxylic acid based styryl/alkyne hybrid molecule as a...
Tác giả: Richa Singh, Vishal M Balaramnavar, Rabi Sankar Bhatta, Amol Chhatrapati Bisen, Anil N Gaikwad, Sanchita Gupta, Nilesh Khandelwal, Ravindra Kumar, Santosh Kumar, Vinita Kushwaha, Prashant Rai, Sumit K Rastogi, Astha Singh, Arun K Sinha, Salil Varshney
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  331.21649
 
Discovery of novel imidazo[1,2-b]pyridazine derivatives as potent covalent inhibitors of CDK12/13
Tác giả: Meng Xia, Hong Ding, Shuangxi Gu, Yongchang He, Linghao Hu, Siqi Huang, Hanrui Jiang, Yuanqing Li, Ziteng Li, Cheng Luo, Lei Tang, Mingliang Wang
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  302.222
 
Design, synthesis, and biological evaluation of β-carboline derivatives as ABCB1 inhibitors for reversing multidrug resi...
Tác giả: Yuanyuan Wang, Zhe Chen, Nanjin Ding, Lianghu Gu, Wen Liu, Weiguang Sun, Fengqing Wang, Yonghui Zhang, Yunpeng Zhao
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  331.21649
 
Discovery of β-amino acid substituted naphthalene sulfonamide derivatives as potent Kelch-like ECH-associated protein 1-...
Tác giả: Ziquan Zhao, Yuxin Ge, Zhengyu Jiang, Hongjin Lu, Mengchen Lu, Junjie Wang, Tingting Wu, Shicheng Xu, Qidong You
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  512.56
 
Discovery of highly potent dual GSPT1/BRD4 degraders with anti-AML activity
Tác giả: Yue Xu, Jianping Cai, Chunhong Chen, Binbin Cheng, Dapeng Dai, Jie Fu, Ruijuan Gao, Chunyi Guo, Yun Hong, Ke Li, Yunxuan Li, Qinrong Lin, Zebei Lu, Yuying Qi, Ningning Shi, Shuanghu Wang, Hang Yang, Jiaming Zhang, Fangling Zhao
Xuất bản: France: European journal of medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  551.456
 

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