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91-100 trong số 142 kết quả
Design, synthesis and biological evaluation of non-glucosidal based 1,3,4-thiadiazoles as SGLT-2 inhibitors
Tác giả: Shivani Sharma, Shubham Kumar, Jeena Gupta, Amit Mittal, Navneet Khurana
Xuất bản: England: Future medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  576.54
 
Design, synthesis, biological evaluation, and mechanism of action of new pyrazines as anticancer agents in vitro and in vivo
Tác giả: Jin-Xia Lan, Le-Jun Huang, Si-Shuang Kang, Hao-Huang, Sheng-Lan Liu, Wei Dai, Xin-Liang Xu, Jin-Yang Wang, Guang-Zhao Shu, Wen Hou
Xuất bản: England: Bioorganic & medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  576.54
 
Design, synthesis and biological evaluation of benzo[b]thiophene analogues as novel ferroptosis inhibitor that inhibit fibrosarcoma cell proliferation
Tác giả: Hua Yang, Mingmei Guo, Sumeng Guan, Yuanyuan Chang, Xiaoya Wu, Yinuo Wang, Ling Zhu, Moran Sun
Xuất bản: England: Bioorganic & medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  004.338
 
Synthesis, design, and cholinesterase inhibitory activity of novel 1,2,4-triazole Schiff bases: A combined experimental and computational approach
Tác giả: Hilal Medetalibeyoğlu, Abdurrahman Atalay, Rüya Sağlamtaş, Sevda Manap, Ahmet Buğra Ortaakarsu, Emel Ekinci, Haydar Yüksek, Burak Tüzün
Xuất bản: Netherlands: International journal of biological macromolecules , 2025
Bộ sưu tập: NCBI
ddc:  662.662
 
Design, synthesis, and biological activity of human glutaminyl cyclase inhibitors against Alzheimer's disease
Tác giả: Jingjing Li, Keli Zong, Chaochun Wei, Qidi Zhong, Hong Yan, Juan Wang, Xingzhou Li
Xuất bản: England: Bioorganic & medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  662.662
 
Design, synthesis, and biological evaluation of novel 3-naphthylthiophene derivatives as potent SIRT2 inhibitors for the treatment of myocardial fibrosis
Tác giả: Zhuo Zhang, Chao Ma, Xiong Gao, Chuncheng Wang, Yanchun Li, Chen Yang, Enlong Ma, Maosheng Cheng
Xuất bản: United States: Bioorganic chemistry , 2025
Bộ sưu tập: NCBI
ddc:  678.72
 
Design, synthesis and biological evaluation of truncated 1'-homologated 4'-selenonucleosides as PPARγ/δ dual modulators
Tác giả: Hongseok Choi, Seungchan An, Young Eum Hyun, Minsoo Noh, Lak Shin Jeong
Xuất bản: United States: Bioorganic chemistry , 2025
Bộ sưu tập: NCBI
ddc:  338.456
 
Design, synthesis and activity evaluation of reduction-responsive anticancer peptide temporin-1CEa drug conjugates
Tác giả: Zhenbin Han, Yue Wang, Wenxuan Wang, Maosheng Cheng, Huali Yang, Yang Liu
Xuất bản: United States: Bioorganic chemistry , 2025
Bộ sưu tập: NCBI
ddc:  338.456
 
Design, synthesis and biological evaluation of novel urolithin derivatives targeting liver cancer cells
Tác giả: Mi Tian, Yu Lan, Chen Li, Yipeng Ling, Lirong Zhao, Benhong Zhou
Xuất bản: England: Journal of enzyme inhibition and medicinal chemistry , 2025
Bộ sưu tập: NCBI
ddc:  745.4
 
Bioactive Indanes: Design, synthesis and bioactivity investigation of 2,2-substituted Indane derivatives, a new bioactive Indane scaffold
Tác giả: Tao Zhang, Kit Chan, Abdulilah Ece, Robin Daly, Aoife Cannon, Gaia A Scalabrino, Neil Frankish, Jacintha O'Sullivan, Padraig Fallon, Helen Sheridan
Xuất bản: United States: Bioorganic chemistry , 2025
Bộ sưu tập: NCBI
ddc:  620.004
 

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